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代谢疾病Novel, potent, selective and cellular active ABC type PTP1B inhibitors containing (methanesulfonyl-phenyl-amino)-acetic acid methyl ester phosphotyrosine mimetic.

期刊:Bioorganic & medicinal chemistry发表年份:2015作者:Peihong Liu; Yongli Du; Lianhua Song; Jingkang Shen; Qunyi Li

代谢疾病Optical Control of Insulin Secretion Using an Incretin Switch.

期刊:Angewandte Chemie (International ed. in English)发表年份:2015作者:Johannes Broichhagen; Tom Podewin; Helena Meyer-Berg; Yorrick von Ohlen; Natalie R Johnston; Ben J Jones; Stephen R Bloom; Guy A Rutter; Anja Hoffmann-Röder; David J Hodson; Dirk Trauner

代谢疾病Role of Δ1-pyrroline-5-carboxylate dehydrogenase supports mitochondrial metabolism and host-cell invasion of Trypanosoma cruzi.

期刊:The Journal of biological chemistry发表年份:2015作者:Brian S Mantilla; Lisvane S Paes; Elizabeth M F Pral; Daiana E Martil; Otavio H Thiemann; Patricio Fernández-Silva; Erick L Bastos; Ariel M Silber

代谢疾病Aminopyrazolo[1,5-a]pyrimidines as potential inhibitors of Mycobacterium tuberculosis: Structure activity relationships and ADME characterization.

期刊:Bioorganic & medicinal chemistry发表年份:2015作者:Candice Soares de Melo; Tzu-Shean Feng; Renier van der Westhuyzen; Richard K Gessner; Leslie J Street; Garreth L Morgans; Digby F Warner; Atica Moosa; Krupa Naran; Nina Lawrence; Helena I M Boshoff; Clifton E Barry; C John Harris; Richard Gordon; Kel