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心血管疾病Discovery of 1-butyl-3-chloro-4-(4-phenyl-1-piperidinyl)-(1H)-pyridone (JNJ-40411813): a novel positive allosteric modulator of the metabotropic glutamate 2 receptor.

期刊:Journal of medicinal chemistry发表年份:2014作者:José María Cid; Gary Tresadern; Guillaume Duvey; Robert Lütjens; Terry Finn; Jean-Philippe Rocher; Sonia Poli; Juan Antonio Vega; Ana Isabel de Lucas; Encarnación Matesanz; María Lourdes Linares; José Ignacio Andrés; Jesús Alcazar; José Manuel Alonso

心血管疾病Structure-activity relationship studies toward the discovery of selective apelin receptor agonists.

期刊:Journal of medicinal chemistry发表年份:2014作者:Jean-François Margathe; Xavier Iturrioz; Rodrigo Alvear-Perez; Claire Marsol; Stéphanie Riché; Hadjila Chabane; Nassera Tounsi; Maxime Kuhry; Denis Heissler; Marcel Hibert; Catherine Llorens-Cortes; Dominique Bonnet

心血管疾病Characterization of the novel positive allosteric modulator, LY2119620, at the muscarinic M(2) and M(4) receptors.

期刊:Molecular pharmacology发表年份:2014作者:Carrie H Croy; Douglas A Schober; Hongling Xiao; Anne Quets; Arthur Christopoulos; Christian C Felder

心血管疾病Activation of fibroblast-like synoviocytes derived from rheumatoid arthritis via lysophosphatidic acid-lysophosphatidic acid receptor 1 cascade.

期刊:Arthritis research & therapy发表年份:2014作者:Yoshishige Miyabe; Chie Miyabe; Yoshiko Iwai; Waka Yokoyama; Chiyoko Sekine; Kazutaka Sugimoto; Masayoshi Harigai; Masayuki Miyasaka; Nobuyuki Miyasaka; Toshihiro Nanki