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药效评价LPK-26, a novel kappa-opioid receptor agonist with potent antinociceptive effects and low dependence potential.

期刊:European journal of pharmacology发表年份:2008作者:Yi-Min Tao; Qing-Lin Li; Cong-Fen Zhang; Xue-Jun Xu; Jie Chen; Ya-Wen Ju; Zhi-Qiang Chi; Ya-Qiu Long; Jing-Gen Liu

药效评价Me-talnetant and osanetant interact within overlapping but not identical binding pockets in the human tachykinin neurokinin 3 receptor transmembrane domains.

期刊:Molecular pharmacology发表年份:2008作者:Pari Malherbe; Caterina Bissantz; Anne Marcuz; Claudia Kratzeisen; Marie-Thérèse Zenner; Joseph G Wettstein; Hasane Ratni; Claus Riemer; Will Spooren

药效评价Optimisation and validation of a medium-throughput electrophysiology-based hNav1.5 assay using IonWorks.

期刊:Journal of pharmacological and toxicological methods发表年份:2008作者:A R Harmer; N Abi-Gerges; A Easter; A Woods; C L Lawrence; B G Small; J-P Valentin; C E Pollard

药效评价Pharmacological characterization of ligands at recombinant NMDA receptor subtypes by electrophysiological recordings and intracellular calcium measurements.

期刊:Combinatorial chemistry & high throughput screening发表年份:2008作者:Kasper B Hansen; Hans Bräuner-Osborne; Jan Egebjerg