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代谢疾病The MCH(1) receptor, an anti-obesity target, is allosterically inhibited by 8-methylquinoline derivatives possessing subnanomolar binding and long residence times.

期刊:British journal of pharmacology发表年份:2014作者:T Sakurai; K Ogawa; Y Ishihara; S Kasai; M Nakayama

代谢疾病Physicochemically and pharmacokinetically stable nonapeptide KISS1 receptor agonists with highly potent testosterone-suppressive activity.

期刊:Journal of medicinal chemistry发表年份:2014作者:Taiji Asami; Naoki Nishizawa; Hisanori Matsui; Yoshihiro Takatsu; Atsuko Suzuki; Atsushi Kiba; Michiko Terada; Kimiko Nishibori; Masaharu Nakayama; Junko Ban; Shin-ichi Matsumoto; Naoki Tarui; Yukihiro Ikeda; Masashi Yamaguchi; Masami Kusaka; Tetsuya

代谢疾病Oral delivery of glucagon like peptide-1 by a recombinant Lactococcus lactis.

期刊:Pharmaceutical research发表年份:2014作者:Payal Agarwal; Pulkit Khatri; Blasé Billack; Woon-Kai Low; Jun Shao

代谢疾病Discovery of selective hexapeptide agonists to human neuromedin U receptors types 1 and 2.

期刊:Journal of medicinal chemistry发表年份:2014作者:Kentaro Takayama; Kenji Mori; Koji Taketa; Akihiro Taguchi; Fumika Yakushiji; Naoto Minamino; Mikiya Miyazato; Kenji Kangawa; Yoshio Hayashi