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代谢疾病C-Glucosides with heteroaryl thiophene as novel sodium-dependent glucose cotransporter 2 inhibitors.

期刊:Bioorganic & medicinal chemistry发表年份:2013作者:Yuichi Koga; Shigeki Sakamaki; Mitsuya Hongu; Eiji Kawanishi; Toshiaki Sakamoto; Yasuo Yamamoto; Hirotaka Kimata; Keiko Nakayama; Chiaki Kuriyama; Yasuaki Matsushita; Kiichiro Ueta; Minoru Tsuda-Tsukimoto; Sumihiro Nomura

代谢疾病Polar transmembrane interactions drive formation of ligand-specific and signal pathway-biased family B G protein-coupled receptor conformations.

期刊:Proceedings of the National Academy of Sciences of the United States of America发表年份:2013作者:Denise Wootten; John Simms; Laurence J Miller; Arthur Christopoulos; Patrick M Sexton

代谢疾病Inhibition of calcitonin gene-related peptide (CGRP) has the potential to extend first-phase insulin secretion.

期刊:Experimental and clinical endocrinology & diabetes : official journal, German Society of Endocrinology [and] German Diabetes Association发表年份:2013作者:H Tanaka; R Kashiwagi; T Koizumi

代谢疾病Phosphatidylethanolamine deficiency in Mammalian mitochondria impairs oxidative phosphorylation and alters mitochondrial morphology.

期刊:The Journal of biological chemistry发表年份:2013作者:Guergana Tasseva; Helin Daniel Bai; Magdalena Davidescu; Alois Haromy; Evangelos Michelakis; Jean E Vance