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心血管疾病Structural sweet spot for A1 adenosine receptor activation by truncated (N)-methanocarba nucleosides: receptor docking and potent anticonvulsant activity.

期刊:Journal of medicinal chemistry发表年份:2012作者:Dilip K Tosh; Silvia Paoletta; Francesca Deflorian; Khai Phan; Steven M Moss; Zhan-Guo Gao; Xiaohui Jiang; Kenneth A Jacobson

心血管疾病Synthesis and evaluation of γ-lactam analogs of PGE₂ as EP4 and EP2/EP4 agonists.

期刊:Bioorganic & medicinal chemistry发表年份:2012作者:Tohru Kambe; Toru Maruyama; Yoshihiko Nakai; Hiroji Oida; Takayuki Maruyama; Nobutaka Abe; Akio Nishiura; Hisao Nakai; Masaaki Toda

心血管疾病Determination of dalcetrapib by liquid chromatography-tandem mass spectrometry.

期刊:Journal of pharmaceutical and biomedical analysis发表年份:2012作者:Katja Heinig; Franz Bucheli; Olaf Kuhlmann; Manfred Zell; Axel Pähler; Elke Zwanziger; Günter Gross; Joseph Tardio; Tomohiro Ishikawa; Tomoko Yamashita

心血管疾病Novel selective allosteric and bitopic ligands for the S1P(3) receptor.

期刊:ACS chemical biology发表年份:2012作者:Euijung Jo; Barun Bhhatarai; Emanuela Repetto; Miguel Guerrero; Sean Riley; Steven J Brown; Yasushi Kohno; Edward Roberts; Stephan C Schürer; Hugh Rosen