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代谢疾病Natural product vindoline stimulates insulin secretion and efficiently ameliorates glucose homeostasis in diabetic murine models.

期刊:Journal of ethnopharmacology发表年份:2013作者:Xin-gang Yao; Fanglei Chen; Ping Li; Lingling Quan; Jing Chen; Liang Yu; Hong Ding; Chenjing Li; Lili Chen; Zhaobing Gao; Ping Wan; Lihong Hu; Hualiang Jiang; Xu Shen

代谢疾病Structure-activity-relationship studies around the 2-amino group and pyridine core of antimalarial 3,5-diarylaminopyridines lead to a novel series of pyrazine analogues with oral in vivo activity.

期刊:Journal of medicinal chemistry发表年份:2013作者:Yassir Younis; Frederic Douelle; Diego González Cabrera; Claire Le Manach; Aloysius T Nchinda; Tanya Paquet; Leslie J Street; Karen L White; K Mohammed Zabiulla; Jayan T Joseph; Sridevi Bashyam; David Waterson; Michael J Witty; Sergio Wittlin; Susan

代谢疾病Treatment with CNX-011-67, a novel GPR40 agonist, delays onset and progression of diabetes and improves beta cell preservation and function in male ZDF rats.

期刊:BMC pharmacology & toxicology发表年份:2013作者:Nagesh Gowda; Anilkumar Dandu; Jaideep Singh; Sanghamitra Biswas; Vijaya Raghav; Mudigere N Lakshmi; Pavagada C Shilpa; Venkategowda Sunil; Ashokkumar Reddy; Manojkumar Sadasivuni; Kumaraswamy Aparna; Mahesh Kumar Verma; Yoganand Moolemath; Mammen O

代谢疾病Hydrogen improves glycemic control in type1 diabetic animal model by promoting glucose uptake into skeletal muscle.

期刊:PloS one发表年份:2013作者:Haruka Amitani; Akihiro Asakawa; Kaichun Cheng; Marie Amitani; Kaori Kaimoto; Masako Nakano; Miharu Ushikai; Yingxiao Li; Minglun Tsai; Jiang-Bo Li; Mutsumi Terashi; Huhe Chaolu; Ryozo Kamimura; Akio Inui