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其他Discovery of 7-oxopyrazolo[1,5-a]pyrimidine-6-carboxamides as potent and selective CB(2) cannabinoid receptor inverse agonists.

期刊:Journal of medicinal chemistry发表年份:2013作者:Mojgan Aghazadeh Tabrizi; Pier Giovanni Baraldi; Giulia Saponaro; Allan R Moorman; Romeo Romagnoli; Delia Preti; Stefania Baraldi; Emanuela Ruggiero; Cristina Tintori; Tiziano Tuccinardi; Fabrizio Vincenzi; Pier Andrea Borea; Katia Varani

其他Allele-specific N-glycosylation delays human surfactant protein B secretion in vitro and associates with decreased protein levels in vivo.

期刊:Pediatric research发表年份:2013作者:Saija Taponen; Johanna M Huusko; Ulla E Petäjä-Repo; Reija Paananen; Susan H Guttentag; Mikko Hallman; Ritva Haataja

其他Core refinement toward permeable β-secretase (BACE-1) inhibitors with low hERG activity.

期刊:Journal of medicinal chemistry发表年份:2013作者:Tobias Ginman; Jenny Viklund; Jonas Malmström; Jan Blid; Rikard Emond; Rickard Forsblom; Anh Johansson; Annika Kers; Fredrik Lake; Fernando Sehgelmeble; Karin J Sterky; Margareta Bergh; Anders Lindgren; Patrik Johansson; Fredrik Jeppsson; Johanna Fäl

其他Proprotein convertases process and thereby inactivate formylglycine-generating enzyme.

期刊:The Journal of biological chemistry发表年份:2013作者:Eva C Ennemann; Karthikeyan Radhakrishnan; Malaiyalam Mariappan; Michaela Wachs; Thomas H Pringle; Bernhard Schmidt; Thomas Dierks