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药效评价Synthesis of new 4-heteroaryl-2-phenylquinolines and their pharmacological activity as NK-2/NK-3 receptor ligands.

期刊:Archiv der Pharmazie发表年份:2007作者:Anna Borioni; Carlo Mustazza; Isabella Sestili; Maria Sbraccia; Luciana Turchetto; Maria Rosaria Del Giudice

药效评价Validation of a rapid, non-radioactive method to quantify internalisation of G-protein coupled receptors.

期刊:Naunyn-Schmiedeberg's archives of pharmacology发表年份:2007作者:Maikel Jongsma; Urszula M Florczyk; Mariëlle C Hendriks-Balk; Martin C Michel; Stephan L M Peters; Astrid E Alewijnse

药效评价Solid phase synthesis and SAR of small molecule agonists for the GPR40 receptor.

期刊:Bioorganic & medicinal chemistry letters发表年份:2007作者:Stephen C McKeown; David F Corbett; Aaron S Goetz; Thomas R Littleton; Eric Bigham; Celia P Briscoe; Andrew J Peat; Steve P Watson; Deirdre M B Hickey

药效评价Synthesis and evaluation of homo-bivalent GnRHR ligands.

期刊:Bioorganic & medicinal chemistry发表年份:2007作者:Kimberly M Bonger; Richard J B H N van den Berg; Laura H Heitman; Ad P IJzerman; Julia Oosterom; Cornelis M Timmers; Herman S Overkleeft; Gijsbert A van der Marel