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药效评价Discovery and characterization of 4'-(2-furyl)-N-pyridin-3-yl-4,5'-bipyrimidin-2'-amine (LAS38096), a potent, selective, and efficacious A2B adenosine receptor antagonist.

期刊:Journal of medicinal chemistry发表年份:2007作者:Bernat Vidal; Arsenio Nueda; Cristina Esteve; Teresa Domenech; Sonia Benito; Raquel F Reinoso; Mercè Pont; Marta Calbet; Rosa López; María Isabel Cadavid; María Isabel Loza; Alvaro Cárdenas; Núria Godessart; Jorge Beleta; Graham Warrellow; Hamish Ryd

药效评价1,5-Biaryl pyrrole derivatives as EP1 receptor antagonists: Structure-activity relationships of 4- and 5-substituted benzoic acid derivatives.

期刊:Bioorganic & medicinal chemistry letters发表年份:2007作者:Adrian Hall; Susan H Brown; Iain P Chessell; Anita Chowdhury; Nicholas M Clayton; Tanya Coleman; Gerard M P Giblin; Beverley Hammond; Mark P Healy; Matthew R Johnson; Ann Metcalf; Anton D Michel; Alan Naylor; Riccardo Novelli; David J Spalding; Jenni

药效评价Old drug, new tricks: the unexpected effect of doxazosin on high-density lipoprotein.

期刊:Circulation research发表年份:2007作者:Alan T Remaley

药效评价Synthesis and SAR of 2-aryl pyrido[2,3-d]pyrimidines as potent mGlu5 receptor antagonists.

期刊:Bioorganic & medicinal chemistry letters发表年份:2007作者:John A Wendt; Susan D Deeter; Susan E Bove; Christopher S Knauer; Rachel M Brooker; Corinne E Augelli-Szafran; Roy D Schwarz; Jack J Kinsora; Kenneth S Kilgore