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药效评价Synthesis of sialic acid derivatives as ligands for the myelin-associated glycoprotein (MAG).

期刊:Bioorganic & medicinal chemistry发表年份:2007作者:Sachin V Shelke; Gan-Pan Gao; Stefanie Mesch; Heiko Gäthje; Soerge Kelm; Oliver Schwardt; Beat Ernst

药效评价Azetidinones as vasopressin V1a antagonists.

期刊:Bioorganic & medicinal chemistry发表年份:2007作者:Christophe D Guillon; Gary A Koppel; Michael J Brownstein; Michael O Chaney; Craig F Ferris; Shi-Fang Lu; Karine M Fabio; Marvin J Miller; Ned D Heindel; David C Hunden; Robin D G Cooper; Stephen W Kaldor; Jeffrey J Skelton; Bruce A Dressman; Michael

药效评价Gatifloxacin induces augmented insulin release and intracellular insulin depletion of pancreatic islet cells.

期刊:Biological & pharmaceutical bulletin发表年份:2007作者:Takashi Tomita; Mariko Onishi; Eiji Sato; Yasuhiro Kimura; Kenji Kihira

药效评价The discovery of 2-anilinothiazolones as 11beta-HSD1 inhibitors.

期刊:Bioorganic & medicinal chemistry letters发表年份:2007作者:Chester Yuan; David J St Jean; Qingyian Liu; Lynn Cai; Aiwen Li; Nianhe Han; George Moniz; Ben Askew; Randall W Hungate; Lars Johansson; Lars Tedenborg; David Pyring; Meredith Williams; Clarence Hale; Michelle Chen; Rod Cupples; Jiandong Zhang; Steve