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药效评价Hybrid approach for the design of highly affine and selective dopamine D(3) receptor ligands using privileged scaffolds of biogenic amine GPCR ligands.

期刊:Bioorganic & medicinal chemistry发表年份:2007作者:Britta C Sasse; Ulrich R Mach; Jukka Leppaenen; Thierry Calmels; Holger Stark

药效评价A heparan sulfate-facilitated and raft-dependent macropinocytosis of eosinophil cationic protein.

期刊:Traffic (Copenhagen, Denmark)发表年份:2007作者:Tan-Chi Fan; Hao-Teng Chang; I-Wen Chen; Hsiu-Yiu Wang; Margaret Dah-Tsyr Chang

药效评价Scouting human A3 adenosine receptor antagonist binding mode using a molecular simplification approach: from triazoloquinoxaline to a pyrimidine skeleton as a key study.

期刊:Journal of medicinal chemistry发表年份:2007作者:Erika Morizzo; Francesca Capelli; Ombretta Lenzi; Daniela Catarzi; Flavia Varano; Guido Filacchioni; Fabrizio Vincenzi; Katia Varani; Pier Andrea Borea; Vittoria Colotta; Stefano Moro

药效评价Partial retro-inverso, retro, and inverso modifications of hydrazide linked bifunctional peptides for opioid and cholecystokinin (CCK) receptors.

期刊:Journal of medicinal chemistry发表年份:2007作者:Yeon Sun Lee; Richard S Agnes; Peg Davis; Shou-wu Ma; Hamid Badghisi; Josephine Lai; Frank Porreca; Victor J Hruby