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代谢疾病Synthesis and biological evaluation of novel C-indolylxylosides as sodium-dependent glucose co-transporter 2 inhibitors.

期刊:European journal of medicinal chemistry发表年份:2012作者:Chun-Hsu Yao; Jen-Shin Song; Chiung-Tong Chen; Teng-Kuang Yeh; Tsung-Chih Hsieh; Szu-Huei Wu; Chung-Yu Huang; Yu-Lin Huang; Min-Hsien Wang; Yu-Wei Liu; Chi-Hui Tsai; Chidambaram Ramesh Kumar; Jinq-Chyi Lee

代谢疾病Synthesis and pharmacological evaluation of indolinone derivatives as novel ghrelin receptor antagonists.

期刊:Bioorganic & medicinal chemistry发表年份:2012作者:Letizia Puleo; Pietro Marini; Roberta Avallone; Marco Zanchet; Silvio Bandiera; Marco Baroni; Tiziano Croci

代谢疾病Rising intracellular zinc by membrane depolarization and glucose in insulin-secreting clonal HIT-T15 beta cells.

期刊:Experimental diabetes research发表年份:2012作者:Kira G Slepchenko; Yang V Li

代谢疾病Discovery of Ipragliflozin (ASP1941): a novel C-glucoside with benzothiophene structure as a potent and selective sodium glucose co-transporter 2 (SGLT2) inhibitor for the treatment of type 2 diabetes mellitus.

期刊:Bioorganic & medicinal chemistry发表年份:2012作者:Masakazu Imamura; Keita Nakanishi; Takayuki Suzuki; Kazuhiro Ikegai; Ryota Shiraki; Takashi Ogiyama; Takeshi Murakami; Eiji Kurosaki; Atsushi Noda; Yoshinori Kobayashi; Masayuki Yokota; Tomokazu Koide; Kazuhiro Kosakai; Yasufumi Ohkura; Makoto Takeuc