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药效评价Pre- and post-Golgi translocation of glucosylceramide in glycosphingolipid synthesis.

期刊:The Journal of cell biology发表年份:2007作者:David Halter; Sylvia Neumann; Suzanne M van Dijk; Jasja Wolthoorn; Ann M de Mazière; Otilia V Vieira; Peter Mattjus; Judith Klumperman; Gerrit van Meer; Hein Sprong

药效评价A monoclonal antibody prevents aggregation of the NBD1 domain of the cystic fibrosis transmembrane conductance regulator.

期刊:Protein engineering, design & selection : PEDS发表年份:2007作者:V Lovato; C Roesli; J Ahlskog; J Scheuermann; D Neri

药效评价ABP688, a novel selective and high affinity ligand for the labeling of mGlu5 receptors: identification, in vitro pharmacology, pharmacokinetic and biodistribution studies.

期刊:Bioorganic & medicinal chemistry发表年份:2007作者:Samuel Hintermann; Ivo Vranesic; Hans Allgeier; Armin Brülisauer; Daniel Hoyer; Michel Lemaire; Thomas Moenius; Stephan Urwyler; Steven Whitebread; Fabrizio Gasparini; Yves P Auberson

药效评价Neurokinin-3 receptor-specific antagonists talnetant and osanetant show distinct mode of action in cellular Ca2+ mobilization but display similar binding kinetics and identical mechanism of binding in ligand cross-competition.

期刊:Molecular pharmacology发表年份:2007作者:Gaochao Tian; Dee Wilkins; Clay W Scott