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代谢疾病Pharmacological profile of ipragliflozin (ASP1941), a novel selective SGLT2 inhibitor, in vitro and in vivo.

期刊:Naunyn-Schmiedeberg's archives of pharmacology发表年份:2012作者:Atsuo Tahara; Eiji Kurosaki; Masanori Yokono; Daisuke Yamajuku; Rumi Kihara; Yuka Hayashizaki; Toshiyuki Takasu; Masakazu Imamura; Li Qun; Hiroshi Tomiyama; Yoshinori Kobayashi; Atsushi Noda; Masao Sasamata; Masayuki Shibasaki

代谢疾病Systematic evaluation of the metabolic to mitogenic potency ratio for B10-substituted insulin analogues.

期刊:PloS one发表年份:2012作者:Tine Glendorf; Louise Knudsen; Carsten E Stidsen; Bo F Hansen; Anne Charlotte Hegelund; Anders R Sørensen; Erica Nishimura; Thomas Kjeldsen

代谢疾病Synthesis, structure-activity relationship, and pharmacological studies of novel melanin-concentrating hormone receptor 1 antagonists 3-aminomethylquinolines: reducing human ether-a-go-go-related gene (hERG) associated liabilities.

期刊:Journal of medicinal chemistry发表年份:2012作者:Shizuo Kasai; Makoto Kamata; Shinichi Masada; Jun Kunitomo; Masahiro Kamaura; Tomohiro Okawa; Kazuaki Takami; Hitomi Ogino; Yoshihide Nakano; Shuntarou Ashina; Kaoru Watanabe; Tomoko Kaisho; Yumi N Imai; Sunghi Ryu; Masaharu Nakayama; Yasutaka Nagisa

代谢疾病Deregulation of CREB signaling pathway induced by chronic hyperglycemia downregulates NeuroD transcription.

期刊:PloS one发表年份:2012作者:In-Su Cho; Miyoung Jung; Ki-Sun Kwon; Eunpyo Moon; Jang-Hyeon Cho; Kun-Ho Yoon; Ji-Won Kim; Young-Don Lee; Sung-Soo Kim; Haeyoung Suh-Kim