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代谢疾病DA-1229, a novel and potent DPP4 inhibitor, improves insulin resistance and delays the onset of diabetes.

期刊:Life sciences发表年份:2012作者:Mi-Kyung Kim; Yu Na Chae; Ha Dong Kim; Eun Kyoung Yang; Eun Jung Cho; Song-hyen Choi; Ye-Hwang Cheong; Hae-Sun Kim; Heung Jae Kim; Yeong Woo Jo; Moon-Ho Son; Soon-Hoe Kim; Chang Yell Shin

代谢疾病Aberrant activation of liver X receptors impairs pancreatic beta cell function through upregulation of sterol regulatory element-binding protein 1c in mouse islets and rodent cell lines.

期刊:Diabetologia发表年份:2012作者:Z X Meng; Y Yin; J H Lv; M Sha; Y Lin; L Gao; Y X Zhu; Y J Sun; X Han

代谢疾病Optimization of co-agonism at GLP-1 and glucagon receptors to safely maximize weight reduction in DIO-rodents.

期刊:Biopolymers发表年份:2012作者:Jonathan W Day; Vasily Gelfanov; David Smiley; Paul E Carrington; George Eiermann; Gary Chicchi; Mark D Erion; Jas Gidda; Nancy A Thornberry; Matthias H Tschöp; Donald J Marsh; Ranabir SinhaRoy; Richard DiMarchi; Alessandro Pocai

代谢疾病Agonism and antagonism at the insulin receptor.

期刊:PloS one发表年份:2012作者:Louise Knudsen; Bo Falck Hansen; Pia Jensen; Thomas Åskov Pedersen; Kirsten Vestergaard; Lauge Schäffer; Blagoy Blagoev; Martin B Oleksiewicz; Vladislav V Kiselyov; Pierre De Meyts