代谢疾病Discovery of a novel glucagon receptor antagonist N-[(4-{(1S)-1-[3-(3, 5-dichlorophenyl)-5-(6-methoxynaphthalen-2-yl)-1H-pyrazol-1-yl]ethyl}phenyl)carbonyl]-β-alanine (MK-0893) for the treatment of type II diabetes.
期刊:Journal of medicinal chemistry发表年份:2012作者:Yusheng Xiong; Jian Guo; Mari R Candelore; Rui Liang; Corey Miller; Qing Dallas-Yang; Guoqiang Jiang; Peggy E McCann; Sajjad A Qureshi; Xinchun Tong; Shiyao Sherrie Xu; Jackie Shang; Stella H Vincent; Laurie M Tota; Michael J Wright; Xiaodong Yang; B