郑州微飒生物科技有限责任公司 咨询热线:0371-88821766
行业动态

行业动态

追踪行业前沿,洞察产业趋势

药效评价Pharmacological characterization of JNJ-28583867, a histamine H(3) receptor antagonist and serotonin reuptake inhibitor.

期刊:European journal of pharmacology发表年份:2007作者:Ann J Barbier; Leah Aluisio; Brian Lord; Ying Qu; Sandy J Wilson; Jamin D Boggs; Pascal Bonaventure; Kirsten Miller; Ian Fraser; Lisa Dvorak; Cindy Pudiak; Christine Dugovic; Jonathan Shelton; Curt Mazur; Michael A Letavic; Nicholas I Carruthers; Tim

药效评价Design and synthesis of novel sulfonamide-containing bradykinin hB2 receptor antagonists. 2. Synthesis and structure-activity relationships of alpha,alpha-cycloalkylglycine sulfonamides.

期刊:Journal of medicinal chemistry发表年份:2007作者:Daniela Fattori; Cristina Rossi; Christopher I Fincham; Valerio Caciagli; Fernando Catrambone; Piero D'Andrea; Patrizia Felicetti; Martina Gensini; Elena Marastoni; Rossano Nannicini; Marielle Paris; Rosa Terracciano; Alessandro Bressan; Sandro Giuli

药效评价2-Aminotetraline derivative protects from ischemia/reperfusion brain injury with a broad therapeutic window.

期刊:Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology发表年份:2007作者:Carmen Capone; Cinzia Fabrizi; Paola Piovesan; Maria Cristina Principato; Patrizia Marzorati; Orlando Ghirardi; Lorenzo Fumagalli; Paolo Carminati; Maria Grazia De Simoni

药效评价A novel multivalent ligand that bridges the allosteric and orthosteric binding sites of the M2 muscarinic receptor.

期刊:Molecular pharmacology发表年份:2007作者:Tod Steinfeld; Mathai Mammen; Jacqueline A M Smith; Richard D Wilson; Jeffrey R Jasper